{"id":242,"date":"2022-10-27T23:43:11","date_gmt":"2022-10-27T21:43:11","guid":{"rendered":"http:\/\/www.congressi.unisi.it\/ewdsy\/?page_id=242"},"modified":"2023-05-12T10:54:17","modified_gmt":"2023-05-12T08:54:17","slug":"programme","status":"publish","type":"page","link":"https:\/\/www.congressi.unisi.it\/ewdsy\/programme\/","title":{"rendered":"Programme"},"content":{"rendered":"\n<p class=\"has-text-align-center\"><strong><u>Sunday 21<sup>st<\/sup> May 2023<\/u><\/strong><\/p>\n\n\n\n<p class=\"has-text-align-left\">14.00 &#8211; 19.00\u2002<em>Registration and posters\u2019 billsticking<\/em><\/p>\n\n\n\n<p class=\"has-text-align-center\"><strong>Sala Bracci &#8211; Certosa di Pontignano &#8211;<\/strong> <strong>Maurizio Botta&#8217;s Friends afternoon<\/strong><\/p>\n\n\n\n<p><em>Opening Remarks:<\/em> <em>Greetings from the Magnificent Rector<\/em> <strong>Prof. Roberto Di Pietra<\/strong><br>17.00\u2002<strong>Welcome Prof. Bruno Botta<\/strong> <em>University of Roma &#8220;La Sapienza&#8221;<\/em> <em>(Italy)<\/em><br>17.15 \u2002<strong>Prof. Stephen Neidle<\/strong> <em>University College London<\/em> <em>(UK)<\/em><br>\u2002\u2002\u2002\u2002\u2002<span style=\"color:#007acc\" class=\"tadv-color\">\u2002A structure-based approach to the design of quadruplex DNA targeting anticancer drugs: <br>\u2002\u2002\u2002\u2002\u2002\u2002identification of a clinical candidate<\/span><br>17.40\u2002<strong>Prof. Karl-Heinz Altmann<\/strong> <em>ETH Z\u00fcrich<\/em><strong> <\/strong><em>(Switzerland)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#007acc\" class=\"tadv-color\">The Chemistry and Biology of (Certain) Macrocyclic Natural Products<\/span><br>18.10\u2002<strong>Prof. Thierry Langer<\/strong> <em>University of Wien<\/em> <em>(Austria)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#007acc\" class=\"tadv-color\">Merging computational and medicinal chemistry: Maurizio Botta as a role model<\/span><br>18.30\u2002<strong>Prof.<\/strong><em> <\/em><strong>Dieter Schinzer<\/strong> <em>University of Magdeburg<\/em> <em>(Germany)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#007acc\" class=\"tadv-color\">Total Synthesis of Biologically Active Natural Products<\/span><\/p>\n\n\n\n<p class=\"has-text-align-left\">19.30\u2002<span style=\"color:#1a1a1a\" class=\"tadv-color\"><em>Dinner<\/em><\/span><br>21.00\u2002Official Opening <strong>Prof. Elena Petricci<\/strong><br>21.15\u2002 <strong>Dr. Rino Rappuoli<\/strong> <em>Biotecnopolo (Italy)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#007acc\" class=\"tadv-color\">Digital Vaccines<\/span><\/p>\n\n\n\n<p class=\"has-text-align-center\"><strong><u>Monday 22<sup>nd<\/sup> May 2023<\/u><\/strong><br><em><strong>Sala Bracci &#8211; Certosa di Pontignano<\/strong><\/em><br><em><strong><span style=\"color:#00a310\" class=\"tadv-color\">Green Chemistry in Drug Synthesis<\/span><\/strong><\/em><\/p>\n\n\n\n<p class=\"has-text-align-left\">09.00\u2002<strong>Dr. Tobias Ritter<\/strong> <em>Max Planck Institut<\/em> <em>(Germany)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#00a310\" class=\"tadv-color\">Late-Stage Functionalizations<\/span><br>09.45\u2002<strong>Prof. Luigi Vaccaro<\/strong> <em>University of Perugia<\/em> <em>(Italy)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#00a310\" class=\"tadv-color\">Sustainability challenges and synthetic tools for target molecules<\/span><br>10.30\u2002 <strong>Prof. Kurt Faber<\/strong> <em>University of Graz<\/em> <em>(Austria)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002 <span style=\"color:#00a310\" class=\"tadv-color\">Biocatalytic API-Synthesis<\/span><\/p>\n\n\n\n<p><em>11.15&nbsp;&nbsp;&nbsp; Coffee break<\/em><\/p>\n\n\n\n<p>11.45\u2002<strong>Prof. Daniele Castagnolo<\/strong> <em>University College London (UK)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#00a310\" class=\"tadv-color\">Biocatalytic and chemo-enzymatic cascades in the synthesis of drug building blocks<\/span><br>12.30\u2002<strong>Prof. Darren Dixon<\/strong> <em>University of Oxford<\/em> <em>(UK)<\/em><br>\u2002\u2002\u2002\u2002\u2002<span style=\"color:#00a310\" class=\"tadv-color\">\u2002New Broad Scope Strategies for Amine Synthesis<\/span><br>13.15\u2002<strong>Dr. Alice Pedruzzi<\/strong> <em>B\u00fcchi<\/em> <em>(Italy)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#00a310\" class=\"tadv-color\">Chromatography with supercritical fluid applied to the preparatory purification technique<\/span><\/p>\n\n\n\n<p><em>13.30\u00a0\u00a0 Lunch<\/em><\/p>\n\n\n\n<p class=\"has-text-align-left\">14.30\u2002<em>Poster session<\/em><\/p>\n\n\n\n<p class=\"has-text-align-center\"><strong>Symeres Afternoon<\/strong><br><strong><span style=\"color:#e746d1\" class=\"tadv-color\">New Synthetic Strategies in Medical Chemistry<\/span><\/strong><\/p>\n\n\n\n<p>15.30\u2002<strong>Dr. Andr\u00e9 De Vries<\/strong><em> <em>Symeres<\/em><\/em> <em>(Netherlands)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#e746d1\" class=\"tadv-color\">Moving towards green chemistry in drug development, why and how<\/span><\/p>\n\n\n\n<p>16.15\u00a0\u00a0\u00a0<em><strong>Symeres &#8211; AXXAM TEAM WORKS<\/strong><\/em><\/p>\n\n\n\n<p><em>17.15\u2002Coffee break<\/em><\/p>\n\n\n\n<p>17.45\u00a0\u00a0\u00a0<em><strong>Symeres &#8211; AXXAM TEAM WORKS<\/strong><\/em><\/p>\n\n\n\n<p>19.30\u2002<em>Dinner<\/em><\/p>\n\n\n\n<p><em>21.00\u2002AFTER DINNER: SYMERES Wine Tasting<\/em><\/p>\n\n\n\n<p class=\"has-text-align-center\"><strong><u>Tuesday 23<sup>rd<\/sup> May 2023<\/u><\/strong><br><strong>Sala Bracci &#8211; Certosa di Pontignano<\/strong><br><em><strong><span style=\"color:#fada0c\" class=\"tadv-color\">New Synthetic Strategies in Medicinal Chemistry<\/span><\/strong><\/em><\/p>\n\n\n\n<p>9.00\u2002<strong>Dr. Anna K.H. Hirsch<\/strong> <em>Helmholtz Centre for Infection Research<\/em> <em>(Germany)<\/em><br>\u2002\u2002\u2002\u2002\u2002 <span style=\"color:#cfb407\" class=\"tadv-color\">Addressing under explored anti-infective drug targets<\/span><br>9.45\u2002<strong>Prof. Maria Laura Bolognesi<\/strong> <em>University of Bologna<\/em> <em>(Italy)<\/em><br>\u2003\u2003  \u00a0<span style=\"color:#cfb407\" class=\"tadv-color\">Sustainable synthesis of drugs and bioactive compounds from food waste<\/span><br>10.30\u2002<strong>Dr. Lloyd Payne<\/strong> <em>Arrepath<\/em> <em>(USA)<\/em><br>\u2003\u2003 \u00a0 <span style=\"color:#cfb407\" class=\"tadv-color\">Harnessing microscopy with machine learning: the search for new classes of antibacterials\u2019<\/span><br>11.15\u2002Oral Communication 1<\/p>\n\n\n\n<p><em>11.35\u2002Coffee break<\/em><\/p>\n\n\n\n<p>11.50\u2002<strong>Dr. Maria Pia Catalani<\/strong> <em>AXXAM (Italy)<\/em><br>\u2002\u2002\u2002\u2002\u2002 <span style=\"color:#cfb407\" class=\"tadv-color\">Hit the road<\/span><br>12.20\u2002<strong>Dr. Phil Cox<\/strong> <em>AbbVie (USA)<\/em><br>\u2003\u2003 \u00a0 <span style=\"color:#cfb407\" class=\"tadv-color\">Computational approaches to drug properties etc. His approach at Abbvie<\/span><br>13.00\u2002Oral Communication 2<br>13.15\u2002 Flash Communication 1<br>13.22\u2002Flash Communication 2<\/p>\n\n\n\n<p><em>13.30&nbsp;&nbsp; Lunch<\/em><\/p>\n\n\n\n<p>14.30\u2002<strong>Dr. Maria Rosaria Romano<\/strong> <em>GSK (Italy)<\/em><br>\u2003\u2003\u2003<span style=\"color:#cfb407\" class=\"tadv-color\">New technologies pave the way for next generation glycoconjugate vaccines<\/span><br>15.00\u2002<strong>Dr. Jacob Bush<\/strong> <em>GSK (UK)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#cfb407\" class=\"tadv-color\">Expanding the liganded proteome with reactive fragments<\/span><br>15.30\u2002<strong>Dr. Louise Walport<\/strong> <em>Crick Institute (UK)<\/em><br>15.55\u2002Oral Communication 3<br>16.10\u2002Flash Communication 3<br>16.17\u2002Flash Communication 4<br>16.25\u2002Flash Communication 5<br>16.32\u2002Flash Communication 6<\/p>\n\n\n\n<p><em><em>16.40\u2002Coffee break<\/em><\/em><\/p>\n\n\n\n<p>16.55\u2002<strong>Dr. Samuele Cazzamalli and <strong>Francesca Migliorini<\/strong><\/strong> <em>Philochem (Switzerland)<\/em><br>\u2002\u2002\u2002\u2002\u2002\u2002<span style=\"color:#cfb407\" class=\"tadv-color\">Drug Discovery with DNA-encoded Libraries (DEL)<\/span><\/p>\n\n\n\n<p><em>20.30\u00a0\u00a0 Bus departure from Certosa di Pontignano to Piazza Gramsci (Siena)<\/em><br><em>20.30\u00a0\u00a0 Social Dinner in Siena<\/em><\/p>\n\n\n\n<p class=\"has-text-align-center\"><strong><u>Wednesday 24<sup>th<\/sup> May 2023<\/u><\/strong><br><strong>Sala Bracci &#8211; Certosa di Pontignano<\/strong><\/p>\n\n\n\n<p>09.00\u2002Oral Communication 4<br>09.15\u2002Oral Communication 5<br>09.30\u2002Oral Communication 6<br>09.45\u2002Flash Communication 7<br>09.52\u2002Flash Communication 8<br>09.59\u2002Flash Communication 9<br>10.06\u2002Flash Communication 10<br>10.13 \u2002Flash Communication 11<br>10.20  Flash Communication 12<br>10.27\u2002<strong><span style=\"color:#007acc\" class=\"tadv-color\">Best poster and Best team works awards<\/span><\/strong><\/p>\n\n\n\n<p><em>10.50\u2002Coffee break<\/em><\/p>\n\n\n\n<p>11.20\u2002<strong><span style=\"color:#007acc\" class=\"tadv-color\">Presentation of best posters and team works<\/span><\/strong><br>12.10\u2002<strong><span style=\"color:#007acc\" class=\"tadv-color\">Closing lecture<\/span><\/strong> <strong>Dr. Russel Thomas<\/strong> <em>Symeres (Netherlands)<\/em><br>\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0<span style=\"color:#007acc\" class=\"tadv-color\">21<sup>st<\/sup> Century drug discovery, challenges and some solutions<\/span><br>12.50\u2002<strong><span style=\"color:#007acc\" class=\"tadv-color\">Closing Remarks<\/span><\/strong> <strong>Prof. Elena Petricci<\/strong><\/p>\n\n\n\n<p><em>13.00\u2002Lunch<\/em><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Sunday 21st May 2023 14.00 &#8211; 19.00\u2002Registration and posters\u2019 billsticking Sala Bracci &#8211; Certosa di Pontignano &#8211; Maurizio Botta&#8217;s Friends afternoon Opening Remarks: Greetings from the Magnificent Rector Prof. Roberto Di Pietra17.00\u2002Welcome Prof. Bruno Botta University of Roma &#8220;La Sapienza&#8221; (Italy)17.15 \u2002Prof. Stephen Neidle University College London (UK)\u2002\u2002\u2002\u2002\u2002\u2002A structure-based approach to the design of quadruplex &hellip; <a href=\"https:\/\/www.congressi.unisi.it\/ewdsy\/programme\/\" class=\"more-link\">Leggi tutto<span class=\"screen-reader-text\"> &#8220;Programme&#8221;<\/span><\/a><\/p>\n","protected":false},"author":2,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"saved_in_kubio":false,"footnotes":""},"class_list":["post-242","page","type-page","status-publish","hentry"],"kubio_ai_page_context":{"short_desc":"","purpose":"general"},"_links":{"self":[{"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/pages\/242","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/users\/2"}],"replies":[{"embeddable":true,"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/comments?post=242"}],"version-history":[{"count":20,"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/pages\/242\/revisions"}],"predecessor-version":[{"id":400,"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/pages\/242\/revisions\/400"}],"wp:attachment":[{"href":"https:\/\/www.congressi.unisi.it\/ewdsy\/wp-json\/wp\/v2\/media?parent=242"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}